Highly efficient and eco-friendly one-pot synthesis of penta substitute pyrrole derivatives under catalyst-free conditions

• Autorzy: Viradiya, D. J. , Baria, B. H. , Kakadiya, R. , Kotadiya, V. C. , Shah, A.
• Języki publikacji: EN

Abstrakty

EN

An eco-friendly and efficient one-pot synthesis of penta-substituted pyrrole derivatives via a four-component reaction of maldrum’s acid, arylglyoxal monohydrate, dimethyl but-2-yne-dioate and amines under catalyst-free conditions in an environmentally friendly medium is described. The simple experimental procedure, catalyst-free reaction conditions, short period of conversion, and excellent yields are the advantages of the present method. Good chemical yields have been achieved without the need for chromatography and recrystallization or other purification methods.

Słowa kluczowe

EN

one-pot synthesis; penta-substituted pyrrole derivatives; multi-component reactions

• Czasopismo: International Letters of Chemistry, Physics and Astronomy
• Rocznik: 2014
• Tom: Vol. 11, iss. 3
• Strony: 257--264
• Opis fizyczny: Bibliogr. 10 poz., tab., wz.

Twórcy

autor

Viradiya, D. J.

• Department of Chemistry (UGC-SAP & DST-FIST Sponsored), Saurashtra University, Rajkot -360005, Gujarat, India National Facility for Drug Discovery Center, Saurashtra University, Rajkot -360005, Gujarat, India,

autor

Baria, B. H.

• Department of Chemistry (UGC-SAP & DST-FIST Sponsored), Saurashtra University, Rajkot -360005, Gujarat, India National Facility for Drug Discovery Center, Saurashtra University, Rajkot -360005, Gujarat, India

autor

Kakadiya, R.

• Department of Chemistry (UGC-SAP & DST-FIST Sponsored), Saurashtra University, Rajkot -360005, Gujarat, India National Facility for Drug Discovery Center, Saurashtra University, Rajkot -360005, Gujarat, India

autor

Kotadiya, V. C.

• Department of Chemistry (UGC-SAP & DST-FIST Sponsored), Saurashtra University, Rajkot -360005, Gujarat, India National Facility for Drug Discovery Center, Saurashtra University, Rajkot -360005, Gujarat, India

autor

Shah, A.

• Department of Chemistry (UGC-SAP & DST-FIST Sponsored), Saurashtra University, Rajkot -360005, Gujarat, India National Facility for Drug Discovery Center, Saurashtra University, Rajkot -360005, Gujarat, India,

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