Anti-edematous and antinociceptive activities of new ureide derivatives in experimental models of inflammation in rats

• Autorzy: Librowski T. , Kubacka M. , Filipek B. , Salat K.
• Języki publikacji: EN

Abstrakty

EN

• Wydawca: -
• Czasopismo: Acta Biologica Cracoviensia. Series Zoologia
• Rocznik: 2010
• Tom: 52
• Opis fizyczny: p.61-66,fig.,ref.

Twórcy

autor

Librowski T.

• Department of Pharmacodynamics, Jagiellonian University, Faculty of Pharmacy, Medical College, Medyczna 9, 30-688 Cracow, Poland

autor

Kubacka M.

• Department of Pharmacodynamics, Jagiellonian University, Faculty of Pharmacy, Medical College, Medyczna 9, 30-688 Cracow, Poland

autor

Filipek B.

• Department of Pharmacodynamics, Jagiellonian University, Faculty of Pharmacy, Medical College, Medyczna 9, 30-688 Cracow, Poland

autor

Salat K.

• Department of Pharmacodynamics, Jagiellonian University, Faculty of Pharmacy, Medical College, Medyczna 9, 30-688 Cracow, Poland

Bibliografia

• ARBUZOV, B.A., FEDOTOVA, N.R., ZOBOVA, N.N., NAZYROVA, A.Z., ANAN’EV, E.V. and S.M. GORBUNOV. 1989. Synthesis, antiinflammatory and analgesic activity of IV-acylureas. Khim. Farm. Zh. 23: 682-683.
• ASGHAR, A.U., HASAN, S.S. and A.E. KING. 2000. The anticonvulsant remacemide and its metabolite AR- R12495AA attenuate spinal synaptic transmission and carrageenan-induced inflammation in the young rat. Eur. J. Pain 4: 97-106.
• BIANCHI, M., RIPAMONTI, C., PALAZZOLO, L., PAZZUCCONI F. and A.E. PANERAI. 1988. Dissociation of the effects of acute chlomipramine on morphine analgesia and plasma concentrations. Arch. Int. Pharmacodyn. Ther. 295: 34- -39.
• BIANCHI, M., ROSSONI, G., SACERDOTE, P., PANERAI, A.E. and F. BERTI. 1995. Carbamazepine exerts anti-inflammatory effects in the rat. Eur. J. Pharmacol. 294: 71—74.
• BIANCHI, M., SACERDOTE, P. and A.E. PANERAI. 1994. Chlomi¬pramine differently affects inflammatory edema and pain in the rat. Pharmacol. Biochem. Behav. 48: 1037- -1040.
• BOSETTI, F., WEERASINGHE, G.R., ROSENBERGER, T.A. and S.I. RAPOPORT. 2003. Valproic acid down-regulates the conversion of arachidonic acid to eicosanoids via cyclooxygenase-1 and -2 in rat brain. J. Neurochem. 85: 690-696.
• CERBAI, G. and G.F. Di PACO. 1961. On some ureides possessing neurosedative activity. Boll. Chim. Farm. 100: 685-691.
• CHITI, W. 1960. New ureides with local anesthetic action. Farmaco Sci. 15: 29-43.
• CRONSTEIN, B.N., MONTESINOS, M.C. and G. WEISSMANN. 1999. Salicylates and sulfasalazine, but not glucocrticoids, inhibit leukocyte accumulation by an adenosine- dependent mechanism that is independent of inhibition of prostaglandin synthesis and pl05 ofNFxB. Proc. Natl. Acad. Sci. 96: 6377-6381.
• DAWOOD, K.M., ABDEL-GAWAD, H., ELLITHEY, M., MOHAMED, H.A. and B. HEGAZI. 2006. Synthesis, anticonvulsant, and anti-inflammatory activities of some new benzofuran- based heterocycles. Arch. Pharm. (Weinheim). 339: 133- -140.
• FLEKHTER, O.B., BOREKO, E.I., NIGMATULLINA, L.R., TRET’IAKOVA, E.V., PAVLOVA, N.I., BALTINA, L.A., NIKOLAEVA, S.N., SAVINOVA, O.V., GALIN, F.Z. and G.A. TOLSTIKOV. 2003. Synthesis and antiviral activity of ureides and carbamates of betulinic acid and its derivatives. Bioorg. Khim. 29: 655-661.
• HAGHIKIA, A., LADAGE, K, HINKEROHE, D., VOLLMAR, P., HEUPEL, K, DERMIETZEL, R. and P.M. FAUSTMANN. 2008. Implications of antiinflammatory properties of the anticonvulsant drug levetiracetam in astrocytes. J. Neurosci. Res. 86: 1781-1788.
• KASSUYA, C.A., SILVESTRE, A.A., REHDER, V.L. and J.B. CALIXTO. 2003. Anti-allodynic and anti-edematogenic properties of the extract and lignans from Phyllanthus amarus in models of persistent inflammatory and neuropathic pain. Eur. J. Pharmacol. 478: 145—153.
• KIM, Y.K., JUNG, H.G., MYINT, A.M., KIM, H. and S.H. PARK. 2007. Imbalance between pro-inflammatory and anti¬inflammatory cytokines in bipolar disorder. J. Affect. Disord. 104: 91—95.
• KOMATSU, T., AWATA, H., SAKAI, Y., INABA, S. and H. YAMAMOTO. 1973. Additional data on an anti-inflammatory agent, ID-955. Arzneim-Forsch. (Drug Res.). 23: 500-503.
• KRUPP, P. and M. WESP. 1975. Inhibition of prostaglandin synthetase by psychotropic drugs. Experientia 31: 330-331.
• LENĉE, P. 1962. A new device for plethysmoscopic measuring of small objects. Arch Int Pharmacodyn. Ther. 136: 237— -240.
• LIBROWSKI, T., KUBACKA, M., MEUSEL, M., SCOLARI, S., MϋLLER, CH.E.andM.Gϋtschow. 2007. Evaluation of anticonvulsant and analgesic effects of benzyl- and benzhydryl ureides. Eur. J. Pharmacol. 559: 138-149.
• MATOTH, I., PINTO, F., SICSIC, C. and T. BRENNER T. 2000. Inhibitory effect of carbamazepine on inflammatory mediators produced by stimulated glial cells. Neurosci. Res. 38: 209-212.
• MCKINNEY M. 2005. Brain cholinergic vulnerability: relevance to behavior and disease. Biochem. Pharmacol. 70: 1115- -1124.
• PAVIA, M.R., LOBBESTAEL, S.J., TAYLOR, C.P., HERSHENSON, F.M. and D.L. MISKELL. 1990. N-phenyl-N’-pyridinylureas as anticonvulsant agents. J. Med. Chem. 33: 854—861.
• RANDALL, L.O. and J.J. SELITTO. 1957. A method for measu¬rement of analgesic activity on inflamed tissue. Arch. Int. Pharmacodyn. Ill: 409-419.
• RAZA, M., DHARIWAL, M.A., AGEEL, A.M. and S. QURESHI. 1996. Evaluation of the antiinflammatory activity of sodium valproate in rats and mice. Gen. Pharmacol. 27: 1395- -1400.
• SAWYNOK, J. and X.J. Liu, X.J. 2003. Adenosine in the spinal cord and periphery: release and regulation of pain. Prog. Neurobiol. 69: 313-340.
• WINTER, C.A., RISLEY, E.A. and G.W. Nuss. 1962. Carrageenin- induced edema in the hind paw of the rat as an assay for anti-inflammatory drugs. Proc. Soc. Exp. Biol. Med. 111: 544-547.

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