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Abstrakty
Series of 2-mercapto-4-(p-aminophenylsulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide Aa-h were synthesized via the biginelli condensation. 2-mercapto-4-amino-6-(aryl)-pyrimidine-5-carboxamide react with p-acetamidophenylsulphonylchloride in the presence of pyridine 2 to form 2-mercapto-4-(p-acetamidophenylsulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide 3. It was treated with diluted HCl under reflux afforded 2-mercapto-4-(p-aminophenylsulphonylamino)-6-(aryl)-pyrimidine-5-carboxamide A a-h. The newly synthesized compounds were characterized by elemental analyses, infrared (IR), 1H NMR and 13 C NMR spectroscopic investigation.
Rocznik
Tom
Strony
168--173
Opis fizyczny
Bibliogr. 11 poz., wz.
Twórcy
autor
- Department of Chemistry, Saurashtra University, Rajkot - 360005, India
autor
- Department of Chemistry, Saurashtra University, Rajkot - 360005, India
autor
- Department of Chemistry, Saurashtra University, Rajkot - 360005, India
autor
- Department of Chemistry, Saurashtra University, Rajkot - 360005, India
autor
- Department of Chemistry, Saurashtra University, Rajkot - 360005, India
autor
- Department of Chemistry, Saurashtra University, Rajkot - 360005, India
Bibliografia
- [1] O. Kappe, Tetrahedron 49 (1993) 6937-6963.
- [2] K. Atwal, C. Rovnyak, J. Schwartz, S. Moreland, A. Hedberg, Z. Gougoutas, F. Malley, M. Floyd, J. Med. Chem. 33 (1990) 1510-1515.
- [3] S. Atwal, N. Swanson, E. Unger, M. Floyd, S. Moreland, A. Hedberg, C. O’Reilly, J. Med. Chem. 34 (1991) 806-811.
- [4] C. Rovnyak, S. Atwal, A. Hedberg, D. Kimball, S. Moreland, Z. Gougoutas, C. O’Reilly, J. Schwartz, M. F. Malley, J. Med. Chem. 35 (1992) 3254-3263.
- [5] C. Barrow, G. Nantermet, G. Selnick, L. Glass, E. Rittle, F. Gilbert, G. Steele, F. Homnick, M. Freidinger, W. Ransom, P. Kling, D. Reiss, P. Broten, W. Schorm, L. Chang, S. O’Malley, V. Olah, D. Ellis, A. Barrish, K. Kassahun, P. Leppert, D. Nagarathnam, C. Forray, J. Med. Chem. 43 (2000) 2703-2718.
- [6] C. O. Kappe, Acc. Chem. Res. 33 (2000) 879-888.
- [7] J. Modha, N. Datta, H. Parekh, II Farmaco 56 (2001) 641.
- [8] P. Zalavadiya, S. Tala, J.Akbari, H. Joshi, Arch. Pharm 342 (2009) 469.
- [9] A. Trivedi, A. Siddiqui, V. Shah, ARKIVOC 2 (2008) 210.
- [10] A. Trivedi, D. Dodiya, N. Ravat, V. Shah, ARKIVOC 11 (2008) 131.
- [11] A. Trivedi, D. Dodiya, J. Surani, H. Mathukia, N. Ravat, V. Shah, Arch. Pharm. 34 (2008) 435.
Typ dokumentu
Bibliografia
Identyfikator YADDA
bwmeta1.element.baztech-79cac3cc-d722-4f05-b8a9-8dec9fa29636