Pharmacological and insect antifeedant activities of some 3-(2,4-dichloro-5-fluorophenyl)-5-(substituted phenyl)-4,5-dihydro-1H-pyrazole-1-carbothioamides

• Autorzy: Thirunarayanan G.
• Języki publikacji: EN

Abstrakty

EN

A series containing twelve titled compounds were synthesized by solvent-free method and their purities were examined by literature procedure. These compounds were subjected to study the pharmacological effects such as antibacterial, antifungal and antioxidant activities and the insect antifeedant activities using Bauer-Kirby disc diffusion method with their bacterial and fungal strains, DPPH radical scavenging and leaf disc bio-assay method with 4th instar larvae Achoea janata L.

Słowa kluczowe

EN

Halo aryl 4,5-dihydro-1H-pyrazole-1-carbothioamides; antibacterial activity; antifungal activity; antioxidant activity; insect antifeedant activity

• Wydawca: Przedsiębiorstwo Wydawnictw Naukowych "DARWIN"
• Czasopismo: International Letters of Chemistry, Physics and Astronomy
• Rocznik: 2014
• Tom: Vol. 18
• Strony: 47--56
• Opis fizyczny: Bibliogr. 37 poz., rys., tab., wz.

Twórcy

autor

Thirunarayanan G.

• Department of Chemistry, Annamalai University, Annamalainagar - 608002, India

Bibliografia

• [1] S. P. Sakthinathan, G. Vanangamudi, G. Thirunarayanan, Spectrochim. Acta. 95A (2012) 693-700.
• [2] S. Sasikala, K. Thirumurthy, P. Mayavel, G. Thirunarayanan, Org. Med. Chem. Lett. (2012) doi:10.1186/2191-2858-2-20
• [3] P. Descacq, A. Nuhrich, M. Capdepuy, G. Devaux, Eur. J. Med. Chem. 25 (1990) 285-290.
• [4] S. Cihat, T. Ayla, S. Selma, Y. Nuran, J. Indian Chem. Soc. 67 (1990) 571-573.
• [5] N. M. Abunada, H. M. Hassaneen, N. G. Kandile, O. A. Miqdad, Molecules. 13 (2008) 1011-1024.
• [6] R. Mishra, A. Siddiqui, A. Rahman, Shaharyar, Chem. Sci. J. (2010) 783-790.
• [7] S. Kumar, S. Bawa S, S. Drabu, R. Kumar, H. Gupta, Recent Patents on Anti-Infective Drug Discovery 4 (2009) 154-163.
• [8] S. A. F. Rostom, Bioorg. Med. Chem. 14 (2006) 6475-6485.
• [9] A. Solankee, S. Solankee, G. Patel, Rasayan J. Chem. 3 (2008) 581-585.
• [10] S. Sahu, M. Banerjee, A. Samantra, C. Behera, Tropical J. Pharm. Res. 7 (2008) 961-968.
• [11] A. Mathew, T. L. Mary Sheeja, T. Arun Kumar,K. Radha, Hygeia. J. D. Med. 3 (2011) 48-56.
• [12] N. Mishra, D. Sasmal, Bioorg. Med. Chem. Lett. 21 (2011) 1969-1973.
• [13] G. Thirunarayanan, V. Renuka, K. G. Sekar, K. Lakshmanan, K. Anbarasu, International Letters of Chemistry, Physics and Astronomy 4 (2014) 66-81.
• [14] G. Thirunarayanan, Q-Science Connect, (2014) DOI: http://dx.doi.org/ 10.5339/ connect. 2014.18
• [15] P. C. Lv, H. Q. Li, J. Sun, Y. Zhou, H. L. Zhu, Bioorg. Med. Chem. 18 (2010) 4606-4614.
• [16] V. S. Patil, S. J.Wadher, N. A. Karande, P. G.Yeole, Int. J. Univ. Pharm. Life. Sci. 1 (2011) 16-22.
• [17] Z. Özdemir, H. B. Kandilci, B. Gümüsef, Ü. Çalis, A. A. Bilgin, Eur. J. Med. Chem. 42 (2007) 373-379.
• [18] J. T. Li, Y.Yin, L. Li, M. X. Sun, Ultrasonics Sonochem. 17 (2010) 11-13.
• [19] R. Gupta, N. Gupta, A. Jain, Indian J. Chem. 49B (2010) 351-355.
• [20] L. Pizzuti, L. A.Piovesan, A. F. C. Flores, F. H. Quina and C. M. P. Pereira, Ultrasonics Sonochem 16 (2009) 728-731.
• [21] R. Chawla, U. Sahoo, A. Arora, P. C. Sharma, V. Radhakrishnan, Acta. Poloniae. Pharm. Drug Res. 67 (2010) 55-61.
• [22] V. M. Patil, K. R. Desai, Arkivoc. 1 (2004) 123-129.
• [23] K. G. Sekar, G. Thirunarayanan, Int. J. Sci. Res. Know. 1(8) (2013) 299-307.
• [24] G. Thirunarayanan, K, G. Sekar, Org. Chem.: An Indian J. 10(1) (2014) 43-52.
• [25] G. Thirunarayanan, K. G. Sekar, International Letters of Chemistry, Physics and Astronomy 10(1) (2013)18-34.
• [26] G. Thirunarayanan, K. Sekar, Q-Science Connect. (2013). DOI http://dx.doi.org/10.5339,2013.18
• [27] G. Thirunarayananm, K. Sekar, Org. Chem: An Indian J. 9(12) (2013) 483-492.
• [28] K. Ranganathan, R. Suresh, G. Vanangamudi, K. Thirumurthy, P. Mayavel, G. Thirunarayanan, Bull. Chem. Soc. Ethiop. 28(2) (2014) 271-288.
• [29] G. Thirunarayanan, International Letters of Chemistry, Physics and Astronomy 5 (2014) 89-98.
• [30] G. Thirunarayanan, P. Mayavel, K. Thirumurthy, S. Dineshkumar, R. Sasikala, P. Nisha, A. Nithyaranjani, European Chem. Bull. 2(9) (2013) 598-605.
• [31] G. Thirunarayanan, K. Ravi, International Letters of Chemistry, Physics and Astronomy 14 (2013) 44-57.
• [32] G. Thirunarayanan, K. G. Sekar, J. Saudi Chem. Soc. (2013). DOI: 10.1016/j.jscs.2013.12.002.
• [33] A. W. Bauer, W. M. M. Kirby, J.C. Sherris, M. Truck, Am. J. Clin. Pathol. 45 (1966) 493-498.
• [34] G. Vanangamudi, M. Subramanian, G. Thirunarayanan, Arabian J. Chem. (2013) DOI: 10.1016/j.arabjc.2013.03.006.
• [35] K. Ranganathan, R. Suresh, D. Kamalakkannan, R. Arulkumaran, R. Sundararajan, S. P. Sakthinathan, S. Vijayakumar, G. Vanangamudi, K. Thirumurthy, P. Mayavel, G. Thirunarayanan, International Letters of Chemistry, Physics and Astronomy 4 (2012) 66-75.
• [36] G. Thirunarayanan, K. G. Sekar, Int. J. Chem. 2(4) (2013) 513-526.
• [37] V. G. Dethler’s, Chemical Insect Attractants and Repellents, Blackistan, Philadelphia. 1947; p. 210.