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2008 | 6 | 4 | 562-568
Tytuł artykułu

Synthesis, characterization and antifungal testing of 3,4-dihydropyrimidin-2(1H)-(thio)ones containing boronic acids and boronate esters

Treść / Zawartość
Warianty tytułu
Języki publikacji
EN
Abstrakty
EN
The addition of formylphenylboronic acid derivatives to thiourea and ethyl acetoacetate proceeds in the presence of an additional Lewis acid catalyst to give the corresponding 3,4-dihydropyrimidin-2(1H)-(thio)ones (Biginelli products) in moderate yield. Compounds were tested for antifungal activity against pure cultures of Aspergillus niger, Aspergillus flavus, Candida albicans and Saccharomyces cerevisiae but, unfortunately, none showed any appreciable activity. [...]
Wydawca

Czasopismo
Rocznik
Tom
6
Numer
4
Strony
562-568
Opis fizyczny
Daty
wydano
2008-12-01
online
2008-10-28
Twórcy
  • Department of Chemistry, Mount Allison University, Sackville, NB, E4L 1G8, Canada
  • Department of Chemistry, Mount Allison University, Sackville, NB, E4L 1G8, Canada
  • Department of Chemistry, Mount Allison University, Sackville, NB, E4L 1G8, Canada
  • Department of Chemistry, Mount Allison University, Sackville, NB, E4L 1G8, Canada
  • Department of Chemistry, Mount Allison University, Sackville, NB, E4L 1G8, Canada
  • Department of Chemistry, Mount Allison University, Sackville, NB, E4L 1G8, Canada
  • Department of Biology, Mount Allison University, Sackville, NB, E4L 1G7, Canada
  • Department of Chemistry, University of New Brunswick, Fredericton, NB, E3B 5A3, Canada
  • Department of Chemistry, Mount Allison University, Sackville, NB, E4L 1G8, Canada, swestcott@mta.ca
Bibliografia
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Typ dokumentu
Bibliografia
Identyfikatory
Identyfikator YADDA
bwmeta1.element.-psjd-doi-10_2478_s11532-008-0064-x
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